Patient info Open main menu

L01E Protein kinase inhibitors, antineoplastic and immunomodulating agents

ATC group of level 3 – pharmacological subgroup · in plain English: targeted cancer medicines (kinase inhibitors)

This site has the patient leaflet or the SPC of 353 medicines in this group and its subgroups.

Place in the ATC classification

  1. L Antineoplastic and immunomodulating agents 1,791 medicines
    1. L01 Antineoplastic agents 1,025 medicines
      1. L01E Protein kinase inhibitors, antineoplastic and immunomodulating agents 353 medicines
        1. L01EA BCR-ABL tyrosine kinase inhibitors 101 medicines
        2. L01EB Epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors 40 medicines
        3. L01EC B-Raf serine-threonine kinase (BRAF) inhibitors 6 medicines
        4. L01ED Anaplastic lymphoma kinase (ALK) inhibitors 14 medicines
        5. L01EE Mitogen-activated protein kinase (MEK) inhibitors 10 medicines
        6. L01EF Cyclin-dependent kinase (CDK) inhibitors 13 medicines
        7. L01EG Mammalian target of rapamycin (mTOR) kinase inhibitors 27 medicines
        8. L01EH Human epidermal growth factor receptor 2 (HER2) tyrosine kinase inhibitors 4 medicines
        9. L01EJ Janus-associated kinase (JAK) inhibitors 18 medicines
        10. L01EK Vascular endothelial growth factor receptor (VEGFR) tyrosine kinase inhibitors 12 medicines
        11. L01EL Bruton's tyrosine kinase (BTK) inhibitors 8 medicines
        12. L01EM Phosphatidylinositol-3-kinase (Pi3K) inhibitors 6 medicines
        13. L01EX Other protein kinase inhibitors 94 medicines

Medicines in the group and its subgroups

MedicineLegal category
Erlotinib Sandoz 25 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Erlotinib Sun 100 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Erlotinib Sun 150 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Erlotinib Sun 25 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Erlotinib Tillomed 100 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Erlotinib Tillomed 150 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Erlotinib Tillomed 25 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Erlotinib Zentiva 100 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Erlotinib Zentiva 150 mg film-coated tablets SPC no longer supplied (L01EB02 erlotinib) –
Erlotinib Zentiva 25 mg film-coated tablets SPC (L01EB02 erlotinib) Prescription only (POM)
Everolimus 10 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus 2.5 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus 5 mg tablets (L01EG02 everolimus) Prescription only (POM)
Everolimus Ethypharm 10 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus Ethypharm 2.5 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus Ethypharm 5 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus Krka 10 mg tablets (L01EG02 everolimus) Prescription only (POM)
Everolimus Krka 2.5 mg tablets (L01EG02 everolimus) Prescription only (POM)
Everolimus Krka 5 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus Mylan 2.5 mg tablets SPC (L01EG02 everolimus) –
Everolimus Sandoz 10 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus Sandoz 2.5 mg tablets (L01EG02 everolimus) Prescription only (POM)
Everolimus Sandoz 5 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus Teva 10 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus Teva 2.5 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Everolimus Teva 5 mg tablets SPC (L01EG02 everolimus) Prescription only (POM)
Finlee 10 mg dispersible tablets SPC (L01EC02 dabrafenib) Prescription only (POM)
Fotivda 1340 micrograms hard capsules SPC (L01EK03 tivozanib) Prescription only (POM)
Fotivda 890 micrograms hard capsules SPC (L01EK03 tivozanib) Prescription only (POM)
Gefitinib 250 mg film-coated tablets SPC (L01EB01 gefitinib) Prescription only (POM)
Gefitinib Accord 250 mg film-coated tablets SPC (L01EB01 gefitinib) Prescription only (POM)
Gefitinib Glenmark 250 mg film-coated tablets SPC (L01EB01 gefitinib) Prescription only (POM)
Gefitinib Mylan 250 mg film-coated tablets (L01EB01 gefitinib) Prescription only (POM)
Gefitinib Sandoz 250 mg film-coated tablets SPC no longer supplied (L01EB01 gefitinib) –
Giotrif 20 mg film-coated tablets SPC (L01EB03 afatinib) Prescription only (POM)
Giotrif 30 mg film-coated tablets SPC (L01EB03 afatinib) Prescription only (POM)
Giotrif 40 mg film-coated tablets SPC (L01EB03 afatinib) Prescription only (POM)
Giotrif 50 mg film-coated tablets SPC no longer supplied (L01EB03 afatinib) –
Glivec 100 mg film-coated tablets (L01EA01 imatinib) Prescription only (POM)
Glivec 400 mg film-coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Ibrance 100 mg film-coated tablets SPC (L01EF01 palbociclib) Prescription only (POM)
Ibrance 100 mg hard capsules not available (L01EF01 palbociclib) –
Ibrance 125 mg film-coated tablets SPC (L01EF01 palbociclib) Prescription only (POM)
Ibrance 125 mg hard capsules not available (L01EF01 palbociclib) –
Ibrance 75 mg film-coated tablets SPC (L01EF01 palbociclib) Prescription only (POM)
Ibrance 75 mg hard capsules SPC no longer supplied (L01EF01 palbociclib) –
Iclusig SPC no longer supplied (L01EA05 ponatinib) –
Iclusig 15 mg film-coated tablets (L01EA05 ponatinib) Prescription only (POM)
Iclusig 30 mg film-coated tablets SPC (L01EA05 ponatinib) Prescription only (POM)
Iclusig 45 mg film-coated tablets SPC no longer supplied (L01EA05 ponatinib) –
Imatinib 100 mg capsules hard SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib 100 mg dispersible tablets (L01EA01 imatinib) Prescription only (POM)
Imatinib 100 mg film-coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib 400 mg capsules hard SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib 400 mg film-coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib 600 mg film-coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib Accord 100 mg film coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib Accord 400 mg film coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib Actavis SPC (L01EA01 imatinib) –
Imatinib Altan 100 mg hard capsules SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib DR. Reddys 100 mg capsules hard SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib DR. Reddys 400 mg capsules hard SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib Grindeks 100 mg hard capsules SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib Koanaa SPC (L01EA01 imatinib) –
Imatinib Milpharm 100 mg film-coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib Teva SPC (L01EA01 imatinib) –
Imatinib Teva 400 mg film-coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Imatinib Tillomed 100 mg film-coated tablets SPC (L01EA01 imatinib) Prescription only (POM)
Imbruvica 140 mg film-coated tablets SPC (L01EL01 ibrutinib) Prescription only (POM)
Imbruvica 140 mg hard capsules SPC no longer supplied (L01EL01 ibrutinib) –
Imbruvica 280 mg film-coated tablets (L01EL01 ibrutinib) Prescription only (POM)
Imbruvica 420 mg film-coated tablets SPC (L01EL01 ibrutinib) Prescription only (POM)
Imbruvica 560 mg film-coated tablets SPC (L01EL01 ibrutinib) Prescription only (POM)
Inlyta SPC (L01EK01 axitinib) Prescription only (POM)
Inlyta 1 mg film-coated tablets SPC (L01EK01 axitinib) Prescription only (POM)
Inlyta 3 mg film-coated tablets SPC (L01EK01 axitinib) Prescription only (POM)
Inlyta 5 mg film-coated tablets SPC (L01EK01 axitinib) Prescription only (POM)
Inlyta 5 mg Fiml-coated tablets (L01EK01 axitinib) Prescription only (POM)
Inlyta 7 mg film-coated tablets SPC (L01EK01 axitinib) Prescription only (POM)
Inrebic 100 mg capsule hard SPC (L01EJ02 fedratinib) Prescription only (POM)
Iressa 250 mg film-coated tablets SPC (L01EB01 gefitinib) Prescription only (POM)
Jakavi 10 mg tablets SPC (L01EJ01 ruxolitinib) Prescription only (POM)
Jakavi 15 mg tablets SPC (L01EJ01 ruxolitinib) Prescription only (POM)
Jakavi 20 mg tablets SPC (L01EJ01 ruxolitinib) Prescription only (POM)
Jakavi 5 mg tablets SPC (L01EJ01 ruxolitinib) Prescription only (POM)
Jakavi 5 mg/ml oral solution SPC (L01EJ01 ruxolitinib) Prescription only (POM)
Kisplyx 10 mg hard capsules SPC (L01EX08 lenvatinib) Prescription only (POM)
Kisplyx 4 mg hard capsules SPC (L01EX08 lenvatinib) Prescription only (POM)
Kisqali 200 mg film-coated tablets SPC (L01EF02 ribociclib) Prescription only (POM)
Koselugo 10 mg hard capsule SPC (L01EE04 selumetinib) Prescription only (POM)
Koselugo 25 mg hard capsules SPC (L01EE04 selumetinib) Prescription only (POM)
Koselugo 5 mg granules in capsule for Opening (L01EE04 selumetinib) Prescription only (POM)
Koselugo 7.5 mg granules in capsule for Opening SPC (L01EE04 selumetinib) Prescription only (POM)
Lenvatinib 10 mg hard capsules SPC (L01EX08 lenvatinib) Prescription only (POM)
Lenvatinib 4 mg hard capsules SPC (L01EX08 lenvatinib) Prescription only (POM)
Lenvatinib Torrent 10 mg hard capsules SPC (L01EX08 lenvatinib) Prescription only (POM)
Lenvima 10 mg hard capsules SPC (L01EX08 lenvatinib) Prescription only (POM)
Lenvima 4 mg hard capsules (L01EX08 lenvatinib) Prescription only (POM)
Lorviqua 100 mg film-coated tablets SPC (L01ED05 lorlatinib) Prescription only (POM)
Lorviqua 25 mg film-coated tablets SPC (L01ED05 lorlatinib) Prescription only (POM)

Sources

  • Patient leaflets and SPCs: the MHRA product information (products.mhra.gov.uk) and the European Medicines Agency (EMA)
  • Active substances, ATC codes and legal categories: the NHS Dictionary of Medicines and Devices (dm+d), NHS Business Services Authority
  • World Health Organization (WHO): ATC/DDD classification, group L01E

Contains public sector information licensed under the Open Government Licence v3.0.

Ask your doctor or pharmacist which medicine is right for you.